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Showing results 1 to 11 of 11
| Issue Date | Title | Author(s) | 2012 | 3-Pyridyl substituted aliphatic cycles as CYP11B2 inhibitors: aromaticity abolishment of the core significantly increased selectivity over CYP1A2. | Yin, Lina; Hu, Qingzhong; Hartmann, Rolf W; Pharmaceutical and Medicinal Chemistry, Saarland University & Helmholtz Institute for Pharmaceutical Research Saarland (HIPS), Saarbrücken, Germany. |
Sep-2011 | Computational investigation of the binding mode of bis(hydroxylphenyl)arenes in 17β-HSD1: molecular dynamics simulations, MM-PBSA free energy calculations, and molecular electrostatic potential maps. | Negri, Matthias; Recanatini, Maurizio; Hartmann, Rolf W; Pharmaceutical and Medicinal Chemistry, Saarland University and Helmholtz Institute for Pharmaceutical Research Saarland (HIPS), Campus C2.3, 66123 Saarbrücken, Germany. |
May-2012 | Design, synthesis and evaluation of novel 16-imidazolyl substituted steroidal derivatives possessing potent diversified pharmacological properties. | Bansal, Ranju; Guleria, Sheetal; Thota, Sridhar; Bodhankar, Subhash L; Patwardhan, Moreshwar R; Zimmer, Christina; Hartmann, Rolf W; Harvey, Alan L; University Institute of Pharmaceutical Sciences, Sector-14, Panjab University, Chandigarh 160014, India. ranju29in@yahoo.co.in |
23-Mar-2012 | Discovery of antagonists of PqsR, a key player in 2-alkyl-4-quinolone-dependent quorum sensing in Pseudomonas aeruginosa. | Lu, Cenbin; Kirsch, Benjamin; Zimmer, Christina; de Jong, Johannes C; Henn, Claudia; Maurer, Christine K; Müsken, Mathias; Häussler, Susanne; Steinbach, Anke; Hartmann, Rolf W; Helmholtz Institute for Pharmaceutical Research Saarland, Campus C2.3, 66123 Saarbrücken, Germany. |
2012 | Hydroxybenzothiazoles as new nonsteroidal inhibitors of 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1). | Spadaro, Alessandro; Negri, Matthias; Marchais-Oberwinkler, Sandrine; Bey, Emmanuel; Frotscher, Martin; Pharmaceutical and Medicinal Chemistry, Saarland University, Saarbrücken, Germany. |
2011 | Serum microRNA-21 as marker for necroinflammation in hepatitis C patients with and without hepatocellular carcinoma. | Bihrer, Verena; Waidmann, Oliver; Friedrich-Rust, Mireen; Forestier, Nicole; Susser, Simone; Haupenthal, Jörg; Welker, Martin; Shi, Ying; Peveling-Oberhag, Jan; Polta, Andreas; von Wagner, Michael; Radeke, Heinfried H; Sarrazin, Christoph; Trojan, Jörg; Zeuzem, Stefan; Kronenberger, Bernd; Piiper, Albrecht; Department of Medicine I, University of Frankfurt/M., Frankfurt, Germany. |
Sep-2011 | Serum miR-122 as a biomarker of necroinflammation in patients with chronic hepatitis C virus infection. | Bihrer, Verena; Friedrich-Rust, Mireen; Kronenberger, Bernd; Forestier, Nicole; Haupenthal, Jörg; Shi, Ying; Peveling-Oberhag, Jan; Radeke, Heinfried H; Sarrazin, Christoph; Herrmann, Eva; Zeuzem, Stefan; Waidmann, Oliver; Piiper, Albrecht; Department of Medicine I, University of Frankfurt/M., Frankfurt, Germany. |
2011 | Structural basis for species specific inhibition of 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1): computational study and biological validation. | Klein, Tobias; Henn, Claudia; Negri, Matthias; Frotscher, Martin; Pharmaceutical and Medicinal Chemistry, Saarland University, Saarbrücken, Germany. |
2011 | Structural basis for species specific inhibition of 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1): computational study and biological validation. | Klein, Tobias; Henn, Claudia; Negri, Matthias; Frotscher, Martin; Pharmaceutical and Medicinal Chemistry, Saarland University, Saarbrücken, Germany. |
Dec-2012 | Synthesis and aromatase inhibitory activity of some new 16E-arylidenosteroids. | Bansal, Ranju; Thota, Sridhar; Karkra, Nalin; Minu, Maninder; Zimmer, Christina; Hartmann, Rolf W; University Institute of Pharmaceutical Sciences, Sector-14, Panjab University, Chandigarh 160 014, India. ranju29in@yahoo.co.in |
6-Jan-2012 | Synthesis and Biological Evaluation of Spiro-δ-lactones as Inhibitors of 17β-Hydroxysteroid Dehydrogenase Type 2 (17β-HSD2) | Xu, Kuiying; Wetzel, Marie; W. Hartmann, Rolf; Marchais-Oberwinkler, Sandrine |
Showing results 1 to 11 of 11
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